ORG 27569

Description

ORG 27569

Org 27569 is a drug which acts as a potent and selective positive allosteric modulator of the cannabinoid CB1 receptor. Studies in vitro suggest that it binds to a regulatory site on the CB1 receptor target, causing a conformational change that increases the binding affinity of CB1 agonists such as CP 55,940, while decreasing the binding affinity of CB1 antagonists or inverse agonists such as rimonabant.

ORG 27569

IUPAC name: 5-chloro-3-ethyl-1H-indole-2-carboxylic acid [2-(4-piperidin-1-yl-phenyl)ethyl]amide

CAS number: 868273-06-7

Formula: C24H28ClN3O

Purity: 99,0% min

Appearance: white powder

The physiological and toxicological properties of this compound are not known. This product is intended for research and forensic purposes.